• Alleviation of nervous tension
• Anxiolytic properties
• Nootropic potential
• Facilitates falling asleep
• GABA analog

Labolic Phenibut is a preparation containing a derivative of γ-aminobutyric acid (GABA). The product has anxiolytic, calming, and nootropic potential.

Phenibut (β-phenyl-γ-aminobutyric acid) is a phenyl derivative of GABA – the primary inhibitory neurotransmitter. The compound was first synthesized in Russia. Phenibut shows agonism to GABA-B receptors, which makes its mechanism of action similar to baclofen, registered as a drug in spastic conditions of various origins. Phenibut has several dozen times weaker activity than baclofen.

Penetration through the blood-brain barrier
Unlike exogenously ingested GABA, Phenibut can cross the blood-brain barrier, which is why it can increase GABA levels in the brain. This results in a stronger effect than supplements containing GABA.

The impact on the GABA-ergic system
Phenibut, stimulating GABA-B receptors, mimics the action of GABA. GABA has an inhibitory effect on the nervous system, which is manifested by the relief of anxiety and stress, sedation, calming down, and reduction of the excessive tension of skeletal muscles.

Positive effect on mood
Phenibut exerts a slight dopaminergic effect, which is often manifested by an improvement of well-being, an increase of the sense of pleasure, and a reduction of social stress. Hence, it is often used by shy people with social anxiety. Nevertheless, note that phenibut has some addictive potential.

Calm, relaxing sleep
Muscle relaxation and reduction of stress levels undoubtedly facilitate falling asleep. Calm and deep sleep is essential for optimal body regeneration, well-being, and high productivity.

In conclusion, Labolic Phenibut is a preparation with strong pharmacological activity, helpful in combating mild stress and anxiety.